Detalhe da pesquisa
1.
A yellow fever virus NS4B inhibitor not only suppresses viral replication, but also enhances the virus activation of RIG-I-like receptor-mediated innate immune response.
PLoS Pathog
; 18(1): e1010271, 2022 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-35061864
2.
"PROTAC" modified dihydroquinolizinones (DHQs) that cause degradation of PAPD-5 and inhibition of hepatitis A virus and hepatitis B virus, in vitro.
Bioorg Med Chem Lett
; 102: 129680, 2024 Apr 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-38428537
3.
4-Oxooctahydroquinoline-1(2H)-carboxamides as hepatitis B virus (HBV) capsid core protein assembly modulators.
Bioorg Med Chem Lett
; 58: 128518, 2022 02 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-34979256
4.
Synthesis of 4-oxotetrahydropyrimidine-1(2H)-carboxamides derivatives as capsid assembly modulators of hepatitis B virus.
Med Chem Res
; 30(2): 459-472, 2021.
Artigo
em Inglês
| MEDLINE | ID: mdl-33456291
5.
Identification of a 3-ß-homoalanine conjugate of brusatol with reduced toxicity in mice.
Bioorg Med Chem Lett
; 30(23): 127553, 2020 12 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-32971261
6.
HBV core protein allosteric modulators differentially alter cccDNA biosynthesis from de novo infection and intracellular amplification pathways.
PLoS Pathog
; 13(9): e1006658, 2017 Sep.
Artigo
em Inglês
| MEDLINE | ID: mdl-28945802
7.
Discovery and Mechanistic Study of Benzamide Derivatives That Modulate Hepatitis B Virus Capsid Assembly.
J Virol
; 91(16)2017 08 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-28566379
8.
A Novel Benzodiazepine Compound Inhibits Yellow Fever Virus Infection by Specifically Targeting NS4B Protein.
J Virol
; 90(23): 10774-10788, 2016 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-27654301
9.
Novel substituted aminothiazoles as potent and selective anti-hepatocellular carcinoma agents.
Bioorg Med Chem Lett
; 26(23): 5819-5824, 2016 12 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-27793566
10.
A cyclin D1 intrinsically disordered domain accesses modified histone motifs to govern gene transcription.
Oncogenesis
; 13(1): 4, 2024 Jan 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-38191593
11.
Design and synthesis of N-alkyldeoxynojirimycin derivatives with improved metabolic stability as inhibitors of BVDV and Tacaribe virus.
Bioorg Med Chem Lett
; 23(14): 4258-62, 2013 Jul 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-23747225
12.
N-Alkyldeoxynojirimycin derivatives with novel terminal tertiary amide substitution for treatment of bovine viral diarrhea virus (BVDV), Dengue, and Tacaribe virus infections.
Bioorg Med Chem Lett
; 23(7): 2172-6, 2013 Apr 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-23453839
13.
Identification of novel tetrahydroquinoxaline derived phenyl ureas as modulators of the hepatitis B virus nucleocapsid assembly.
Eur J Med Chem
; 259: 115634, 2023 Nov 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-37499290
14.
The Renaissance of CDK Inhibitors in Breast Cancer Therapy: An Update on Clinical Trials and Therapy Resistance.
Cancers (Basel)
; 14(21)2022 Nov 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-36358806
15.
Hepatoselective Dihydroquinolizinone Bis-acids for HBsAg mRNA Degradation.
ACS Med Chem Lett
; 12(7): 1130-1136, 2021 Jul 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-34267883
16.
Identification of hepatitis B virus core protein residues critical for capsid assembly, pgRNA encapsidation and resistance to capsid assembly modulators.
Antiviral Res
; 191: 105080, 2021 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-33933516
17.
Downregulation of histone methyltransferase SET8 inhibits progression of hepatocellular carcinoma.
Sci Rep
; 10(1): 4490, 2020 03 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-32161353
18.
Targeting the multifunctional HBV core protein as a potential cure for chronic hepatitis B.
Antiviral Res
; 182: 104917, 2020 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-32818519
19.
Quassinoid analogs with enhanced efficacy for treatment of hematologic malignancies target the PI3Kγ isoform.
Commun Biol
; 3(1): 267, 2020 05 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-32461675
20.
Discovery of Novel Hepatitis B Virus Nucleocapsid Assembly Inhibitors.
ACS Infect Dis
; 5(5): 759-768, 2019 05 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-30525438